Table 5. PK parameters for in vivo tissue distribution (%ID/g) of the Technekitty injection (Tc-99m)

Organs Tmax (hr) Cmax (%ID/g) AUClast (hr × [%ID/g]) AUCINF_obs (hr × [%ID/g]) CI_obs ({mCi}/{hr × [%ID/g]}/kg) MRTlast (hr) MRTINF_obs (hr) HL_Lambda_z1) (hr)
Blood 0.083 8.358 27.084 28.104 0.024 6.015 6.940 5.198
Heart 0.083 2.780 10.404 11.102 0.060 6.719 8.360 6.108
Liver 0.083 4.903 40.590 67.839 0.010 9.963 26.455 18.730
Lung 0.083 5.447 19.832 21.161 0.032 6.663 8.312 6.189
Spleen 0.083 3.015 10.743 11.456 0.058 6.697 8.330 6.195
Kidney 0.083 4.027 27.515 36.251 0.018 9.150 16.957 12.161
Stomach 2 26.376 298.465 345.810 0.002 8.638 12.349 8.141
Small intestine 1 5.118 33.882 38.890 0.017 8.111 11.735 8.496
Large intestine 6 8.986 124.702 170.379 0.004 10.361 19.308 13.680
Thyroid 2 22.641 211.414 227.777 0.003 7.455 9.282 6.158
Salivary gland 2 25.517 223.304 240.129 0.003 7.419 9.191 6.040
Muscle 0.083 1.049 4.263 4.485 0.149 6.820 8.090 5.931
Femur 0.083 2.411 8.754 9.318 0.072 6.567 8.154 6.108
Brain 0.083 0.256 1.332 1.427 0.469 7.336 9.074 6.589
Testis 0.083 1.224 7.554 8.415 0.080 7.438 10.225 7.418
Terminal half-life of the drug.
ID, injected dose.